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Donepezil Hydrochloride (E2020) and Other Acetylcholinesterase Inhibitors

[ Vol. 7 , Issue. 3 ]

Author(s):

Hachiro Sugimoto, Yoshiharu Yamanish, Youichi Iimura and Yoshiyuki Kawakami   Pages 303 - 339 ( 37 )

Abstract:


A wide range of evidence shows that acetylcholinesterase (AChE) inhibitors can

Keywords:

donepezil hydrochloride,acetylcholinesterase inhibitors,alzheimer s disease,AChE inhibitors,cortical cholinergic neurotransmission,hepatotxic liability,physostigmine,cholineric enhancement therapy,ACh releasers,M1 M3 Receptor agonists,nicotinic agonists,velnacrine,amiridine,eptastigmine,galanthamine,rivastigmine,metrifonate,huperzine A,donepezil hydrocloride,anti AChE Activity,n alkyl analogs,molecular modeling,receptor dependent docking,crystal structure,BuChE,Brain acetylcholine concentrations,TAK 147,anti inflammatory agents,alzheimer s disease treatment,estrogen replacement therapy,anti oxidants,anti amyloid,galanin receptor antagonist

Affiliation:

, , , Tsukuba ResearchLaboratories, Eisai Co., Ltd., 5-1-3 Tokodai, Tsukuba, Ibaraki 300-2635, Japan



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