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Improved, High Yield Synthesis of 3H-Quinazolin-4-ones, the Key Intermediates of Recently Developed Drugs

[ Vol. 11 , Issue. 19 ]

Author(s):

Laszlo Orfi, Frigyes Waczek, Janos Pato, Istvan Varga, Balint Hegymegi-Barakonyi, Richard A. Houghten and Gyorgy Ker   Pages 2549 - 2553 ( 5 )

Abstract:


Purine bases and their bioisosteric analogs are widely used as building blocks in combinatorial chemistry. Recently a great number of fused pyrimidine derivatives became known as potential drug molecules against various types of proliferative diseases, caused by over-expression of protein kinases [1]. One of the most important compound

Keywords:

pyrimidines,quinazolin-4-ones,formamidine-acetate,imidoyl-chlorides,purine analogs,protein kinase inhibitors,antiproliferative agents,phosphodiesterase v inhibitors

Affiliation:

, , , , , , Department of Pharmaceutical Chemistry, Semmelweis University, Hogyes E. u. 9, Budapest, Hungary.



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